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Ʊ³ǹ߱ġῡǴ¾̴١̿ 5ξ˷ϴ½ǵ̶ҸȰϰִ١ ƱDZ Ʊ 25 mg, 50 mg, 100 mgǼٸ̿Ҽִ١½ǵʱ꿰̰ο̿⼺λĮũνīνƮƸ긶׳θν̻ȭƼŸ磬ƮƼƾϰִ١ ǵȭȮ ǵ۵ ǵѹ̹߱߱⸦ϰϴ°´١̾ PDE5ȿۿνۿϴµ PDE5 cGMPcyclic guanosine monophosphate¹ϴ¿Ѵ١ cGMPȰѱ̿ϽŰǰ귯ϴº̴١ ڱµȣü濡ϻȭңNOѴ١ NO cGMPϴ±ƴҷƮŬ̽ҸȿҸȰȭŲ١ PDE5¹߱ӽðϴ cGMPѴ١ǵ PDE5Ͽ cGMPǰ߱ӽðȴ١ Ʊȿ Ʊȿ Ʊ¼ 30п 1ðѴ١Ʊȿºϴ¿뷮 45ðӵȴ١Ʊ½ι߱⸦Űʱ߱⸦̷ؼ¼ڱʿϴ١ Ʊ´索ȯپѿοߵǴ¹߱ġῡȿִ°γŸ١ӻ迡Ʊ¹߱ 80%߱⸦ϰϴ´ɷ۰ι١ Ʊ Ʊӻ Ʊӻ߱ġῡȿߴ١ѿƱѳ 74%ѳ 13%ع߱ⰡǾٰߴ١Ǵٸѳ 25%غƱ߱ 82%ȿ̶°־١ Ʊ½Űջҷι߱Ұɼ̳索ȯڵ鿡ԵǾ١索ִ³ѿƱ¹߱ 59%ȿ־磬ѳ 13%ȿ־١ ƱǺۿ ƱϹ߰ߵٸκۿųִ١ƱǰϹκۿδµ룬ȸȫŻִ١Ѻۿδ帴ѽ÷£ǺȭڸԵȴ١幰ԺƱڱ÷Ұųûִ١ ȯ꿰̳ϴ³ϰԶֱƱؼ¾ȵȴ١ɰѰ̳ȯƯ鵵Ʊϴ°ؾѴ١ƱϱǻͻϿϰȮϴ°߿ϴ١ Ʊۿڼ˾ƺŬ
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Ʊ θ ˷ Դϴ. 1998 ̱ FDA , ӻ ȿ Ǿϴ. ۿ Ʊ ֽ ȿ մϴ.
Ʊ ΰ?
Ʊ ֿ ǵ Ʈ꿰Դϴ. ġ ߵǾ, ۿ ߱ ȿ ߰ߵǸ鼭 ġ DZ ߽ϴ. ߱ ġḦ ǥ Ǿǰ ڸ ҽϴ.
Ʊ ֿ а ۿ Ŀ
ǵ PDE5(-5) ۿմϴ. ڱ ǿ кǴ ϻȭ(NO) ȿ , ظü Ȱ ̿ϰ ŵϴ. ̷ ߱Ⱑ , ߱ ϴ մϴ.
Ʊ ȿ Ǵ
, 80% ߱ ȿ ˴ϴ. Ϲ 30-60 ĺ ȿ Ÿ, 4-5ð ӵ˴ϴ. ڱ ۿϹǷ, ڵ ߱⸦ ʽϴ. ϴ մϴ.
ǻװ ۿ
꿰 迭 (Ʈα۸ ) Բ ؼ ˴ϴ. , ȸ ȫ, ȭҷ, ڸ ۿ ֽϴ. 幰 ÷ ȭ ߱() Ƿ ؾ մϴ.
Ʊ ؿ
Ʊ Ű ƴմϴ. ų ʽϴ. ص Ư ȿ , ݵ ǻ ó濡 ؾ մϴ.
Ű: Ʊ, ǵ, ߱ ġ, PDE5 , , ǰ
ǰ Ʊ ý ǻ
Ʊ Ǹ Ʊ Ʊ þ˸ Ʊ Ʊ
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